Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,081
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1,095
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results
1,081
Tocris Bioscience™ BTZO 1
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CAS: 99420-15-2 Molecular Formula: C13H8N2OS
| CAS | 99420-15-2 |
|---|---|
| Molecular Formula | C13H8N2OS |
1,082
Tocris Bioscience™ TH 5427 Hydrochloride
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Potent NUDT5 inhibitor
| Purity | 98% |
|---|---|
| Chemical Name or Material | 7-[[5-(3,4-Dichlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-1,3-dimethyl-8-(piperazine-1-yl)-1H-purine-2,6-dione hydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C20H20Cl2N8O3.HCl |
| Formula Weight | 527.79 |
1,083
Tocris Bioscience™ Ivabradine hydrochloride
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HCN channel blocker; inhibits If pacemaker current
| CAS | 148849-67-6 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 3-[3-[[[(7S)-3,4-Dimethoxybicyclo[4.2.0]octa-1,3,5-trien-7-yl]methyl]methylamino]propyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-2H-3-benzazepin-2-one hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H36N2O5.HCl |
1,084
Tocris Bioscience™ Pomalidomide 4'-PEG5-amine
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Cereblon ligand with PEG linker and terminal amine for onward chemistry
1,085
Tocris Bioscience™ Megestrol Acetate
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CAS: 595-33-5 Molecular Formula: C24H32O4
| CAS | 595-33-5 |
|---|---|
| Molecular Formula | C24H32O4 |
1,086
Tocris Bioscience™ Rosuvastatin calcium
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Potent HMG-CoA reductase inhibitor
| Target | HMG-CoA Reductase Inhibitors |
|---|---|
| CAS | 147098-20-2 |
| Purity | 99% |
| Chemical Name or Material | (3 R,5 S,6 E)-7-[4-(4-Fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidin-5-yl])-3,5-dihydroxyhept-6-enoic acid hemicalcium salt |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C22H27FN3O6S.1⁄2Ca |
| Formula Weight | Observed MW: 500.57 |
| Assay Percent Range | >99% |
1,087
Tocris Bioscience™ JH-II-127
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Potent and selective LRRK2 inhibitor
| CAS | 1700693-08-8 |
|---|---|
| Chemical Name or Material | [4-[[5-Chloro-4-(methylamino)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxyphenyl]-4-morpholinyl-methanone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H21ClN6O3 |
| Formula Weight | Observed MW: 416.87 |
| Assay Percent Range | >98% |
1,088
Tocris Bioscience™ SCH 202676 hydrobromide
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CAS: 265980-25-4 Molecular Formula: C15H14BrN3S
| CAS | 265980-25-4 |
|---|---|
| Molecular Formula | C15H14BrN3S |
1,089
Tocris Bioscience™ Tiotidine
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CAS: 69014-14-8 Molecular Formula: C10H16N8S2
| CAS | 69014-14-8 |
|---|---|
| Molecular Formula | C10H16N8S2 |
1,090
Tocris Bioscience™ BromoTag™ cis-AGB1
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Negative control for BromoTag AGB1 (Cat.No. 7686)
1,091
Tocris Bioscience™ Gilteritinib
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Potent FLT3 inhibitor; also potently inhibits AXL
| Target | Flt-3/Flk-2/CD135 |
|---|---|
| CAS | 1254053-43-4 |
| Purity | 0.98 |
| Chemical Name or Material | 6-Ethyl-3-[[3-methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]amino]-5-[(tetrahydro-2H-pyran-4-yl)amino]-2-pyrazinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C29H44N8O3 |
1,092
Tocris Bioscience™ AM 580
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CAS: 102121-60-8 Molecular Formula: C22H25NO3
| CAS | 102121-60-8 |
|---|---|
| Molecular Formula | C22H25NO3 |
1,093
Tocris Bioscience™ O4I2
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Oct3/4 inducer; induces expression of pluripotent-associated genes
| Target | Additional Stem Cell Dedifferentiation Products |
|---|---|
| CAS | 165682-93-9 |
| Purity | >98% |
| Chemical Name or Material | Ethyl 2-[(4-chlorophenyl)amino]-4-thiazolecarboxylate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C12H11ClN2O2S |
| Formula Weight | 282.75 |
1,094
Tocris Bioscience™ Ex 26
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Potent and selective S1P1 receptor antagonist
| CAS | 144678-63-7 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Color | White |
| Solubility | Soluble to 100mM in DMSO and to 100mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | 1-[[[5'-[[1-(4-Chloro-3-methylphenyl)ethyl]amino]-2'-fluoro-3,5-dimethyl[1,1'-biphenyl]-4-yl]carbonyl]amino]-cyclopropanecarboxylic acid |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C28H28ClFN2O3 |
| Formula Weight | 494.98 |
1,095
Tocris Bioscience™ PF 04449613, >98%
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CAS: 1236858-52-8 Molecular Formula: C21H25N5O3
| CAS | 1236858-52-8 |
|---|---|
| Molecular Formula | C21H25N5O3 |